Comment
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Synonyms: ,-Dimethyl-4-[2-methyl-8-[2-(3-pyridinyl)ethynyl]-1H-imidazo[4,5-c]quinolin-1-yl]-benzeneacetonitrile A potent, ATP-competitive, dual PI3K/PDK-1 inhibitor in vitro and in vivo (IC = 56, 444, 34, 117 and 240 nM for PI3K p110- ,d, , and PDK1 kinases, respectively). Displays anticancer properties
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